(+)-Enitociclib, CAS 1610358-56-9

Product Description: (+)-Enitociclib ((+)-BAY-1251152) is an enanthiomer of BAY-1251152 with rotation (+). Enitociclib is a potent and selective CDK9 inhibitor with an IC50 of 3 nM. Enitociclib has anti-tumour activity[1][2].

Applications: Cancer-Kinase/protease

Formula: C19H18F2N4O2S

References: [1]Ulrich LÜCKING, et al. 5-fluoro-n-(pyridin-2-yl)pyridin-2-amine derivatives containing a sulfoximine group. WO2014076091A1./[2]Use of Arne Scholz, et al. 5-fluoro-4-(4-fluoro-2-methoxyphenyl)-n-{4-[(s-methylsulfonimidoyl)methyl]pyridin-2-yl}pyridin-2-amine for treating diffuse large b-cell lymphoma. WO2019158517A1.

CAS Number: 1610358-56-9

Molecular Weight: 404.43

Compound Purity: 99.73

Research Area: Cancer

Solubility: DMSO : 113.3 mg/mL (ultrasonic;warming)

Target: CDK

• SKU: MEXHY-103019-10.1
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-103019-10.1
• Package Unit: 10 mM/1 ml
• Quantity Unit: STK