EPZ011989, CAS 1598383-40-4

Product Description: EPZ011989 is a potent and orally active Zeste Homolog 2 (EZH2) inhibitor with metabolic stability. EPZ011989 has inhibitory inhibition for EZH2 with a Ki value of [1]. EPZ011989 is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.

Applications: Cancer-programmed cell death

Formula: C35H51N5O4

References: [1]Campbell JE, et al. EPZ011989, A Potent, Orally-Available EZH2 Inhibitor with Robust in Vivo Activity. ACS Med Chem Lett. 2015 Mar 4;6(5):491-495.

CAS Number: 1598383-40-4

Molecular Weight: 605.81

Compound Purity: 98.79

Research Area: Cancer

Solubility: DMSO : 100 mg/mL (ultrasonic)

Target: Histone Methyltransferase

• SKU: MEXHY-16986-10.1
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-16986-10.1
• Package Unit: 10 mM/1 ml
• Quantity Unit: STK