ERK-MYD88 interaction inhibitor 1, CAS 2215927-89-0

ERK-MYD88 interaction inhibitor 1, CAS 2215927-89-0
SKU
MEXHY-162863-25
Packaging Unit
25 mg
Manufacturer
MedChemExpress

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Product Description: ERK-MYD88 interaction inhibitor 1 is an ERK-MYD88 interaction inhibitor. ERK-MYD88 interaction inhibitor 1 can induce an HRI-mediated integrated stress response (ISR), leading to cancer cell-specific immunogenic cell apoptosis (apoptosis). ERK-MYD88 interaction inhibitor 1 can induce anti-tumor T cell responses in Lewis lung cancer mice, exhibiting anti-tumor activity[1].

Formula: C22H21N5O2

References: [1]Virard F, et al. Targeting ERK-MYD88 interaction leads to ERK dysregulation and immunogenic cancer cell death. Nat Commun. 2024 Aug 15;15(1):7037.

CAS Number: 2215927-89-0

Molecular Weight: 387.43

Compound Purity: 99.02

Research Area: Cancer

Solubility: DMSO : 125 mg/mL (ultrasonic)

Target: Apoptosis
More Information
SKU MEXHY-162863-25
Manufacturer MedChemExpress
Manufacturer SKU HY-162863-25
Package Unit 25 mg
Quantity Unit STK
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