Product Description: ETP-46321 is a potent and orally bioavailable PI3Kα and PI3Kδ inhibitor with Kiapps of 2.3 and 14.2 nM, respectively.
Applications: Cancer-Kinase/protease
Formula: C20H27N9O3S
References: [1]Martínez González S, et al. Identification of ETP-46321, a potent and orally bioavailable PI3K α, δ inhibitor. Bioorg Med Chem Lett. 2012 May 15;22(10):3460-6.
CAS Number: 1252594-99-2
Molecular Weight: 473.55
Compound Purity: 99.34
Research Area: Cancer
Solubility: DMSO : ≥ 33 mg/mL
Target: PI3K