Shelf life (days): 1460.0
Formulation: A solid
Formal Name: (1R,2S)-N-[(cyclopentyloxy)carbonyl]-3-methyl-L-valyl-(4R)-4-[[8-bromo-7-methoxy-2-[2-[(2-methyl-d3-1-oxopropyl)amino-3,3,3-d3]-4-thiazolyl]-4-quinolinyl]oxy]-L-prolyl-1-amino-2-ethenyl-cyclopropanecarboxylic acid
Purity: ≥99% deuterated forms (d1-d2)
Formula Markup: C40H43BrD6N6O9S
Formula Weight: 875.85846
CAS Number: 2750534-88-2
Notes: Faldaprevir-d6 is intended for use as an internal standard for the quantification of faldaprevir by GC- or LC-MS. Faldaprevir is an inhibitor of hepatitis C virus (HCV) non-structural protease 3/4A (NS3/4A; IC50 = 3 nM for the HCV genotype 1b enzyme).{18743} It inhibits genotype 1a and 1b HCV RNA replication in replicon assays (EC50s = 6.5 and 3.1 nM, respectively).{52708}