GB-88, CAS 1416435-96-5

Product Description: GB-88 is an oral, selective non-peptide antagonist of PAR2, inhibits PAR2 activated Ca2+ release with an IC50 of 2 μM[1].

Applications: COVID-19-immunoregulation

Formula: C32H42N4O4

References: [1]Suen JY, et al. Modulating human proteinase activated receptor 2 with a novel antagonist (GB88) and agonist (GB110). Br J Pharmacol. 2012 Mar;165(5):1413-23.

CAS Number: 1416435-96-5

Molecular Weight: 546.70

Compound Purity: 99.05

Research Area: Inflammation/Immunology

Solubility: DMSO : 31.25 mg/mL (ultrasonic)

Target: Protease Activated Receptor (PAR)

• SKU: MEXHY-120261-10.1
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-120261-10.1
• Package Unit: 10 mM/1 ml
• Quantity Unit: STK