GSK0660, CAS 1014691-61-2

Shelf life (days): 1460.0

Formulation: A crystalline solid

Formal Name: 3-[[[2-methoxy-4-(phenylamino)phenyl]amino]sulfonyl]-2-thiophenecarboxylic acid, methyl ester

Purity: ≥95%

Formula Markup: C19H18N2O5S2

Formula Weight: 418.5

CAS Number: 1014691-61-2

Notes: GSK0660 is the first reported antagonist of PPARβ/δ (IC50 = 155 nM) with no measurable affinity for PPARα or PPARγ (IC50s ≥ 10 μM).{32576} Because of the limited bioavailability of GSK0660, the related compound GSK3787 (Item No. 15219) was developed as a selective PPARβ/δ antagonist with more suitable pharmacokinetic properties.{24665}

• SKU: CAY15272-5
• Manufacturer: Cayman Chemical
• Manufacturer SKU: 15272-5
• Package Unit: 5 mg
• Quantity Unit: STK