GSK2807 (Trifluoroacetate), CAS 2245255-66-5

Product Description: GSK2807 Trifluoroacetate is a potent, selective and SAM-competitive inhibitor of SMYD3, with a Ki of 14 nM and an IC50 of 130 nM[1][2].

Formula: C21H33F3N8O7

References: [1]Van Aller GS, et al. Structure-Based Design of a Novel SMYD3 Inhibitor that Bridges the SAM-and MEKK2-Binding Pockets. Structure. 2016 May 3;24(5):774-781./[2]Kaniskan HÜ, et al. Inhibitors of Protein Methyltransferases and Demethylases. Chem Rev. 2018 Feb 14;118(3):989-1068.

CAS Number: 2245255-66-5

Molecular Weight: 566.53

Compound Purity: 99.36

Research Area: Others

Solubility: DMSO : 100 mg/mL (ultrasonic)/H2O : ≥ 50 mg/mL

Target: Histone Methyltransferase

• SKU: MEXHY-104009A-25
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-104009A-25
• Package Unit: 25 mg
• Quantity Unit: STK