HA-130, CAS 1229652-21-4

Shelf life (days): 1460.0

Formulation: A crystalline solid

Formal Name: B-[3-[[4-[[3-[(4-fluorophenyl)methyl]-2,4-dioxo-5-thiazolidinylidene]methyl]phenoxy]methyl]phenyl]-boronic acid

Purity: ≥98%

Formula Markup: C24H19BFNO5S

Formula Weight: 463.3

CAS Number: 1229652-21-4

Notes: HA-130 is a reversible inhibitor of autotaxin, completely blocking the hydrolysis of the substrate bis-pNPP with an IC50 value of 28 nM.{18138} It does not affect the activity of any proteasomal protease or related enzymes. HA-130 rapidly decreases plasma lysophosphatidic acid levels in mice when given intravenously (1 nM/g).{18138} HA-130 has been used to investigate the role of autotaxin in cells and animals.{31823,31824,31825}

• SKU: CAY10498-5
• Manufacturer: Cayman Chemical
• Manufacturer SKU: 10498-5
• Package Unit: 5 mg
• Quantity Unit: STK