Product Description: HIF-2α-IN-1 is a HIF-2α inhibitor with an IC50 value of less than 500 nM.
Applications: Metabolism-sugar/lipid metabolism
Formula: C16H8F5NO4S
References: [1]Bruick Richard Keith, et al. HIF-2α inhibitors for treating iron overload disorders. From PCT Int. Appl. (2016), WO 2016057242 A1 20160414./[2]Dixon Darryl David, et al. Preparation of cyclic sulfone and sulfoximine analogs as HIF-2α inhibitors. From PCT Int. Appl. (2015), WO 2015095048 A1 20150625.
CAS Number: 1799948-06-3
Molecular Weight: 405.30
Compound Purity: 99.92
Research Area: Metabolic Disease
Solubility: DMSO : 100 mg/mL (ultrasonic)
Target: HIF/HIF Prolyl-Hydroxylase