Itriglumide, CAS 201605-51-8

Product Description: Itriglumide (CR 2945) is an anthranilic acid derivative. Itriglumide is a potent and selective CCKB receptor antagonist, with an IC50 of 2.3 nM. Itriglumide antagonizes the response to gastrin in a dose-dependent manner with an IC50 of 5.9 nM. Itriglumide shows antisecretory and antiulcer activity[1].

Applications: COVID-19-immunoregulation

Formula: C33H38N2O4

References: [1]Makovec F, et al. Characterization of antisecretory and antiulcer activity of CR 2945, a new potent and selective gastrin/CCK(B) receptor antagonist. Eur J Pharmacol. 1999 Mar 12;369(1):81-90.

CAS Number: 201605-51-8

Molecular Weight: 526.67

Research Area: Inflammation/Immunology

Target: Cholecystokinin Receptor

• SKU: MEXHY-106347-10
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-106347-10
• Package Unit: 10 mg
• Quantity Unit: STK