K-Ras-PDEδ-IN-1, CAS 1841464-21-8

Product Description: K-Ras-PDEδ-IN-1 is a novel and potent competitive K-Ras-PDEδ inhibitor. K-Ras-PDEδ-IN-1 binds to the farnesyl binding pocket of PDEδ with a low nanomolar Kd of 8 nM[1].

Applications: Cancer-programmed cell death

Formula: C25H26FN5O2

References: [1]Sandip Murarka, et al. Development of Pyridazinone Chemotypes Targeting the PDEδ Prenyl Binding Site. Chemistry. 2017 May 2;23(25):6083-6093.

CAS Number: 1841464-21-8

Molecular Weight: 447.50

Compound Purity: 99.62

Research Area: Cancer

Solubility: DMSO : 12.5 mg/mL (ultrasonic)

Target: Phosphodiesterase (PDE)

• SKU: MEXHY-115555-10.1
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-115555-10.1
• Package Unit: 10 mM/1 ml
• Quantity Unit: STK