L-798,106, CAS 244101-02-8

Shelf life (days): 1460.0

Formulation: A crystalline solid

Formal Name: (2E)-N-[(5-bromo-2-methoxyphenyl)sulfonyl]-3-[2-(2-naphthalenylmethyl)phenyl]-2-propenamide

Purity: ≥95%

Formula Markup: C27H22BrNO4S

Formula Weight: 536.4

CAS Number: 244101-02-8

Notes: Prostaglandin E2 (Item No. 14010) exerts its effects through four separate G-protein coupled receptors (EP1, EP2, EP3, and EP4).{1422} L-798,106 is a highly selective EP3 receptor antagonist with Ki values of 0.3, 916, >5,000, and >5,000 nM at EP3, EP4, EP1, and EP2, respectively.{9826} At 0.2 µM, it blocks the EP3 agonist activity of sulprostone (Item No. 14765) on guinea pig vas deferens and trachea.{26175}

• SKU: CAY11129-5
• Manufacturer: Cayman Chemical
• Manufacturer SKU: 11129-5
• Package Unit: 5 mg
• Quantity Unit: STK