​(Lys5,MeLeu9,Nle10)-Neurokinin A (4-10) (trifluoroacetate s

Shelf life (days): 1460.0

Formulation: A solid

Formal Name: L-a-aspartyl-L-lysyl-L-phenylalanyl-L-valylglycyl-N-methyl-L-leucyl-L-norleucinamide, trifluoroacetate salt

Amino Acids: DKFVG-methyl-LX-NH2 (X = Norleucine)

Purity: ≥98%

Formula Markup: C39H65N9O9 / XCF3COOH

Formula Weight: 804.003

Notes: An NK2 receptor agonist; binds to NK2 receptors in isolated human circular muscle membranes in a radioligand binding assay (IC50 = 0.87 nM); induces contraction of isolated rat bladder and fundus strips (EC50s = 10 and 117 nM, respectively), effects that can be inhibited by the NK2 receptor antagonists SR48968 and MEN10627; induces contraction of uterine horns isolated from rats in proestrus/estrus and diestrus/metestrus (EC50s = 25.12 and 51.29 nM, respectively); induces urination and defecation in conscious dogs but also induces emesis and hypotension at similar doses

• SKU: CAY43051-50
• Manufacturer: Cayman Chemical
• Manufacturer SKU: 43051-50
• Package Unit: 50 mg
• Quantity Unit: STK