Product Description: MC-Val-Cit-PAB-Exatecan (MC-Val-Cit-PAB-DX8951) is a agent-linker conjugate for ADC. MC-Val-Cit-PAB-Exatecan is composed of a DNA topoisomerase I DX-8951 (HY-13631) and a cathepsin cleavable ADC linker.
Applications: Cancer-programmed cell death
Formula: C53H60FN9O12
References: [1]Anish Thomas, et al. Antibody-drug conjugates for cancer therapy. Lancet Oncol. 2016 Jun;17(6):e254-e262.
CAS Number: 2504068-28-2
Molecular Weight: 1034.10
Compound Purity: 99.57
Research Area: Cancer
Solubility: DMSO : 50 mg/mL (ultrasonic)
Target: Drug-Linker Conjugates for ADC;Topoisomerase