Product Description: Olmutinib (HM61713; BI-1482694) is an orally active and irreversible third EGFR tyrosine kinase inhibitor that binds to a cysteine residue near the kinase domain. Olmutinib is used for NSCLC[1][2].
Applications: Cancer-Kinase/protease
Formula: C26H26N6O2S
References: [1]Kim ES, et al. Olmutinib: First Global Approval. Drugs. 2016 Jul;76(11):1153-7./[2]Mohamed W. Attwa, et al. Detection and characterization of olmutinib reactive metabolites by LC‐MS/MS: Elucidation of bioactivation pathways. Journal of Separation science. 18 November 2019.