Perlapine, CAS 1977-11-3

Shelf life (days): 1460.0

Formulation: A crystalline solid

Formal Name: 6-(4-methyl-1-piperazinyl)-11H-dibenz[b,e]azepine

Purity: ≥98%

Formula Markup: C19H21N3

Formula Weight: 291.4

CAS Number: 1977-11-3

Notes: Perlapine is an atypical neuroleptic that blocks dopamine and serotonin (5-HT) receptors (Kis = 60, 30, and 30 nM for D2, D4, and 5-HT2A, respectively).{24252} Perlapine is also an agonist for hM3Dq, a designer receptor exclusively activated by designer drugs (DREADDs) derived from the human muscarinic acetylcholine M3 receptor that activates neuronal firing.{30413} Perlapine displays >10,000-fold selectivity for hM3Dq over hM3.{30413}

• SKU: CAY17756-10
• Manufacturer: Cayman Chemical
• Manufacturer SKU: 17756-10
• Package Unit: 10 mg
• Quantity Unit: STK