PF-05105679, CAS 1398583-31-7

Product Description: PF-05105679 is an orally active and selective TRPM8 antagonist with an IC50 of 103 nM. PF-05105679 has the potential for cold-related pain[1].

Applications: Neuroscience-Neuromodulation

Formula: C26H21FN2O3

References: [1]Andrews MD, et al. Discovery of a Selective TRPM8 Antagonist with Clinical Efficacy in Cold-Related Pain. ACS Med Chem Lett. 2015 Jan 30;6(4):419-24.

CAS Number: 1398583-31-7

Molecular Weight: 428.45

Compound Purity: 99.84

Research Area: Neurological Disease

Solubility: DMSO : 125 mg/mL (ultrasonic)

Target: TRP Channel

• SKU: MEXHY-115506-50
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-115506-50
• Package Unit: 50 mg
• Quantity Unit: STK