Propyl pyrazole triol, CAS 263717-53-9

Propyl pyrazole triol, CAS 263717-53-9
SKU
MEXHY-100689-10.1
Packaging Unit
10 mM/1 ml
Manufacturer
MedChemExpress

Availability: loading...
Price is loading...
Product Description: Propyl pyrazole triol (PPT) is a selective estrogen receptor alpha (ERα) agonist. The relative binding affinity of Propyl pyrazole triol for ERα (ERα: 49%) around 410 times higher compared with estrogen receptor beta (ERβ: 0.12%)[1][2].

Applications: Cancer-programmed cell death

Formula: C24H22N2O3

References: [1]Influence of cellular ERalpha/ERbeta ratio on the ERalpha-agonist induced proliferation of human T47D breast cancer cells./[2]Stauffer SR, et al. Pyrazole ligands: structure-affinity/activity relationships and estrogen receptor-alpha-selective agonists. J Med Chem. 2000 Dec 28;43(26):4934-47.

CAS Number: 263717-53-9

Molecular Weight: 386.44

Compound Purity: 99.11

Research Area: Cancer

Solubility: DMSO : ≥ 100 mg/mL

Target: Estrogen Receptor/ERR
More Information
SKU MEXHY-100689-10.1
Manufacturer MedChemExpress
Manufacturer SKU HY-100689-10.1
Package Unit 10 mM/1 ml
Quantity Unit STK
Product information (PDF) Download
MSDS (PDF) Download