Raltegravir (potassium salt), CAS 871038-72-1

Raltegravir (potassium salt), CAS 871038-72-1
SKU
CAY16071-10
Packaging Unit
10 mg
Manufacturer
Cayman Chemical

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Shelf life (days): 1460.0

Formulation: A crystalline solid

Formal Name: N-[(4-fluorophenyl)methyl]-1,6-dihydro-5-hydroxy-1-methyl-2-[1-methyl-1-[[(5-methyl-1,3,4-oxadiazol-2-yl)carbonyl]amino]ethyl]-6-oxo-4-pyrimidinecarboxamide, monopotassium salt

Purity: ≥98%

Formula Markup: C20H20FN6O5 / K

Formula Weight: 482.5

CAS Number: 871038-72-1

Notes: Raltegravir is an orally bioavailable inhibitor of HIV-1 integrase (IC50 = 15 nM in a strand transfer assay).{26192} It inhibits the spread of HIV-1IIIb infection in MT-4 cell culture with 95% cell culture inhibitory concentration (CIC95) values of 19 and 31 nM in medium containing 10% heat-inactivated fetal bovine serum (FBS) or 50% normal human serum, respectively. Formulations containing raltegravir have been used in combination therapy in the treatment of HIV-1 infection.
More Information
SKU CAY16071-10
Manufacturer Cayman Chemical
Manufacturer SKU 16071-10
Package Unit 10 mg
Quantity Unit STK
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