Elvitegravir-d6

Product Description: Elvitegravir-d6 (GS-9137-d6) is deuterium labeled Elvitegravir. Elvitegravir (GS-9137; JTK-303; D06677) is an HIV integrase inhibitor for HIV-1IIIB, HIV-2EHO and HIV-2ROD with IC50 of 0.7 nM, 2.8 nM and 1.4 nM, respectively[1].

Formula: C23H17D6ClFNO5

References: [1]Russak EM, et al. Impact of Deuterium Substitution on the Pharmacokinetics of Pharmaceuticals. Ann Pharmacother. 2019 Feb;53(2):211-216./[2]Shimura K, et al. Broad antiretroviral activity and resistance profile of the novel human immunodeficiency virus integrase inhibitor elvitegravir (JTK-303/GS-9137). J Virol. 2008 Jan;82(2):764-74.

Molecular Weight: 453.92

Research Area: Infection

Target: HIV;HIV Integrase;Isotope-Labeled Compounds

• SKU: MEXHY-14740S1-0
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-14740S1-0
• Package Unit: Get quote
• Quantity Unit: STK