Enasidenib-d6, CAS 2095569-76-7

Enasidenib-d6, CAS 2095569-76-7
SKU
MEXHY-18690S-1
Packaging Unit
1 mg
Manufacturer
MedChemExpress

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Product Description: Enasidenib-d6 (AG-221-d6) is the deuterium labeled Enasidenib (HY-18690)[1]. Enasidenib is an oral, potent, reversible, selective inhibitor of the IDH2 mutant enzymes, with IC50s of 100 and 400 nM against IDH2R140Q and IDH2R172K, respectively[2].

Formula: C19H11D6F6N7O

References: [1]Russak EM, et al. Impact of Deuterium Substitution on the Pharmacokinetics of Pharmaceuticals. Ann Pharmacother. 2019 Feb;53(2):211-216.

CAS Number: 2095569-76-7

Molecular Weight: 479.41

Research Area: Others

Solubility: 10 mM in DMSO

Target: Isocitrate Dehydrogenase (IDH);Isotope-Labeled Compounds
More Information
SKU MEXHY-18690S-1
Manufacturer MedChemExpress
Manufacturer SKU HY-18690S-1
Package Unit 1 mg
Quantity Unit STK
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