Etbicyphat-13C3

Product Description: Etbicyphat-13C3 is the 13C labeled Etbicyphat (HY-139145). Etbicyphat is a potent GABA(A) receptors competitive antagonist. Etbicyphat induces epileptiform activities in hippocampal CA1 neurons, and binds to the GABA(A)-benzodiazepine receptors[1][2].

Formula: C3 13C3H11O4P

References: [1]Russak EM, et al. Impact of Deuterium Substitution on the Pharmacokinetics of Pharmaceuticals. Ann Pharmacother. 2019 Feb;53(2):211-216./[2]Rijal SO, et al. Dissociation constants for GABA(A) receptor antagonists determined with neuronal networks on microelectrode arrays. J Neurosci Methods. 2008 Aug 30;173(2):183-92.

Molecular Weight: 181.10

Research Area: Neurological Disease

Solubility: 10 mM in DMSO

Target: GABA Receptor

• SKU: MEXHY-139145S-1
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-139145S-1
• Package Unit: 1 mg
• Quantity Unit: STK