S 8849-1-d4 (free base), CAS 1330822-91-7

Product Description: S 8849-1-d4 (free base) (Tianeptine metabolite MC5-d4) is deuterium labeled S 8849-1 (free base). S 8849-1 (free base) (Tianeptine metabolite MC5) is a Tianeptine (HY-90003) metabolite that is found in plasma. The mean elimination half-lives of S 8849-1 (free base) is 7.53 h in rats. S 8849-1 (free base) is promising for research of antidepressants[1][2].

Applications: Neuroscience-Neuromodulation

Formula: C19H17D4ClN2O4S

References: [1]Russak EM, et al. Impact of Deuterium Substitution on the Pharmacokinetics of Pharmaceuticals. Ann Pharmacother. 2019;53(2):211-216./[2]Gaulier JM, et al. High-performance liquid chromatographic determination of tianeptine in plasma applied to pharmacokinetic studies. J Chromatogr B Biomed Sci Appl. 2000 Oct 10;748(2):407-14. /[3]Szafarz M, et al. Pharmacokinetic study of tianeptine and its active metabolite MC5 in rats following different routes of administration using a novel liquid chromatography tandem mass spectrometry analytical method. Naunyn Schmiedebergs Arch Pharmacol. 2018 Feb;391(2):185-196.

CAS Number: 1330822-91-7

Molecular Weight: 412.92

Research Area: Neurological Disease

Target: Drug Metabolite;Isotope-Labeled Compounds

• SKU: MEXHY-166341S-0
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-166341S-0
• Package Unit: Get quote
• Quantity Unit: STK