Tiagabine-d4

Product Description: Tiagabine-d4 (NO050328-d4) is deuterium labeled Tiagabine. Tiagabine (NO050328) is a potent and selective GABA reuptake inhibitor, used as an anticonvulsant agent, with IC50s of 67, 446 and 182 nM for [3H]GABA uptake in Synaptosomes, Neurons and Glia, respectively[1].

Applications: Neuroscience-Neuromodulation

Formula: C20H21D4NO2S2

References: [1]Russak EM, et al. Impact of Deuterium Substitution on the Pharmacokinetics of Pharmaceuticals. Ann Pharmacother. 2019;53(2):211-216.

Molecular Weight: 379.57

Research Area: Neurological Disease

Target: Isotope-Labeled Compounds

• SKU: MEXHY-B0696S1-0
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-B0696S1-0
• Package Unit: Get quote
• Quantity Unit: STK