Toremifene-d6 (hydrochloride)

Product Description: Toremifene-d6 (Z-Toremifene-d6) hydrochloride is deuterium labeled Toremifene. Toremifene is a second-generation selective estrogen-receptor modulator (SERM) in development for the prevention of osteoporosis. Toremifene also potent inhibits infectious EBOV Zaire and Marburg (MARV) with IC50 of 0.07 µM and 2.6 µM, respectively[1][2].

Applications: COVID-19-immunoregulation

Formula: C26H23D6Cl2NO

References: [1]Russak EM, et al. Impact of Deuterium Substitution on the Pharmacokinetics of Pharmaceuticals. Ann Pharmacother. 2019;53(2):211-216./[2]Matthew R Smith, Selective Estrogen Receptor Modulators to Prevent Treatment-Related Osteoporosis.Rev Urol. 2005; 7(Suppl 3): S30-S35.

Molecular Weight: 448.46

Research Area: Infection

Solubility: 10 mM in DMSO

Target: Estrogen Receptor/ERR;Isotope-Labeled Compounds

• SKU: MEXHY-B0005S1-1
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-B0005S1-1
• Package Unit: 1 mg
• Quantity Unit: STK