Product Description: Urapidil-d4 is the deuterium labeled Urapidil[1]. Urapidil is an α1 adrenoreceptor antagonist and a 5-HT1A receptor agonist[2].
Applications: Metabolism-protein/nucleotide metabolism
Formula: C20H25D4N5O3
References: [1]Russak EM, et al. Impact of Deuterium Substitution on the Pharmacokinetics of Pharmaceuticals. Ann Pharmacother. 2019 Feb;53(2):211-216./[2]Bopp C, et al. The effect of urapidil, an alpha-1 adrenoceptor antagonist and a 5-HT1A agonist, on the vascular tone of the porcine coronary and pulmonary arteries, the rat aorta and the human pulmonary artery. Eur J Pharmacol. 2016 May 15;779:53-8.
CAS Number: 1795122-12-1
Molecular Weight: 391.50
Research Area: Endocrinology
Solubility: DMSO : 25 mg/mL (ultrasonic;warming)
Target: 5-HT Receptor;Adrenergic Receptor;Isotope-Labeled Compounds