M871 (trifluoroacetate salt)

Shelf life (days): 1460.0

Formulation: A solid

Formal Name: L-tryptophyl-L-threonyl-L-leucyl-L-asparaginyl-L-seryl-L-alanylglycyl-L-tyrosyl-L-leucyl-L-leucylglycyl-L-prolyl-L-a-glutamyl-L-histidyl-L-prolyl-L-prolyl-L-prolyl-L-alanyl-L-leucyl-L-alanyl-L-leucyl-L-alaninamide, trifluoroacetate salt

Amino Acids: WXLNSAGYLLGPEHPPPALALA-NH2 (X = ξ-threonine)

Purity: ≥95%

Formula Markup: C108H163N27O28 / XCF3COOH

Formula Weight: 2287.615

Notes: A peptide antagonist of GAL2 receptors (Ki = 13.1 nM); selective for GAL2 receptors over GAL1 receptors (Ki = 420 nM); inhibits galanin-induced increases in inositol levels in CHO cells expressing human GAL2 receptors at 0.1, 1, or 10 nM; increases blood glucose, IL-8, IL-6, IL-22, and Tnf-α levels and decreases skeletal muscle and adipocyte Glut4 and Pgc-1α levels in a rat model of diabetes induced by a high-fat diet and STZ when administered intracerebroventricularly

• SKU: CAY42403-1
• Manufacturer: Cayman Chemical
• Manufacturer SKU: 42403-1
• Package Unit: 1 mg
• Quantity Unit: STK