Shelf life (days): 1460.0
Formulation: A solid
Formal Name: 3-[4-(4-amino-1-piperidinyl)-3-(3,5-difluorophenyl)-6-quinolinyl]-2-hydroxy-benzonitrile
Purity: ≥98%
Formula Markup: C27H22F2N4O
Formula Weight: 456.5
CAS Number: 2172870-89-0
Notes: An SST2 agonist; selectively inhibits cAMP production in cells expressing SST2 over cells expressing SST1, SST3, SST4, or SST5 (EC50s = 25, >1,000, >1,000, >1,000, and >1,000 nM, respectively); reduces GHRH-stimulated growth hormone release in rats at 3, 10, and 30 mg/kg; reduces plasma levels of IGF-1 in beagle dogs