BET/Aurora kinase-IN-1, CAS 2674064-32-3

BET/Aurora kinase-IN-1, CAS 2674064-32-3
SKU
MEXHY-170812-0
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MedChemExpress

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Product Description: BET/Aurora kinase-IN-1 (Compound 38) is a dual BET/Aurora kinase inhibitor. BET/Aurora kinase-IN-1 shows antiproliferative activities on diverse cancer cell lines and favorable antitumor efficacy in renal cell cancer and colon cancer xenograft models with tumor growth inhibition (TGI) of 45.99% and 53.06%, respectively[1].

Formula: C25H30FN7O

References: [1]Lyu K, et al. Structure-Based Rational Design and Evaluation of BET-Aurora Kinase Dual-Inhibitors for Treatment of Cancers. J Med Chem. 2025 Jan 23;68(2):1344-1364.

CAS Number: 2674064-32-3

Molecular Weight: 463.55

Research Area: Cancer

Target: Aurora Kinase
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SKU MEXHY-170812-0
Manufacturer MedChemExpress
Manufacturer SKU HY-170812-0
Package Unit Get quote
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