BRD4-BD1-IN-2, CAS 2761321-26-8

Product Description: BRD4-BD1-IN-2 is a selective BRD4-BD1 inhibitor, with an IC50 of 2.51 µM (20-times greater than that of BD2). BRD4-BD1-IN-2 can be used in studies of cancer and cardiovascular diseases[1].

Applications: Cancer-programmed cell death

Formula: C20H15Br3N4O2

References: [1]Chang Y, et al. Design, synthesis, biological evaluation, and molecular docking of 1, 7-dibenzyl-substituted theophylline derivatives as novel BRD4-BD1-selective inhibitors. Medicinal Chemistry Research, 2021, 30(8): 1453-1468.

CAS Number: 2761321-26-8

Molecular Weight: 583.07

Research Area: Cancer; Cardiovascular Disease

Solubility: 10 mM in DMSO

Target: Epigenetic Reader Domain

• SKU: MEXHY-143300-10
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-143300-10
• Package Unit: 10 mg
• Quantity Unit: STK