Casein kinase 1δ-IN-28, CAS 1095750-94-9

Casein kinase 1δ-IN-28, CAS 1095750-94-9
SKU
MEXHY-171278-0
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MedChemExpress

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Product Description: Casein kinase 1δ-IN-28 (Compound 4) is the inhibitor for CK1ε with an IC50 of 0.0146 μM. Casein kinase 1δ-IN-28 exhibits a metabolite rate in human liver microsomes of 52%[1].

Formula: C23H23FN6

References: [1]Vaz RJ, et al., Decreasing the CYP2D6 contribution to metabolism of a CK1ε inhibitor. Bioorg Med Chem Lett. 2018 Dec 15;28(23-24):3681-3684.

CAS Number: 1095750-94-9

Molecular Weight: 402.47

Research Area: Cancer; Metabolic Disease

Target: Casein Kinase
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SKU MEXHY-171278-0
Manufacturer MedChemExpress
Manufacturer SKU HY-171278-0
Package Unit Get quote
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