Cav 3.1 blocker 1, CAS 2158201-04-6

Product Description: Cav 3.1 blocker 1 (compound 12) is a T-type calcium channel blocker with an IC50value of 160 nM for Cav3.1. Cav 3.1 blocker 1 weakly inhibits Cav 3.2 (IC50 of 5000 nM), and shows no inhibition on Cav 3.3 and Cav 1.2 (IC50 of >10000 nM)[1].

Formula: C26H19F6N3O2

References: [1]Bezençon O, et al. Milestones to the Discovery of T-type Calcium Channel Blockers for the Treatment of Generalized Epilepsies. Chimia (Aarau). 2017 Oct 25;71(10):722-729.

CAS Number: 2158201-04-6

Molecular Weight: 519.44

Research Area: Neurological Disease

Target: Calcium Channel

• SKU: MEXHY-156889-0
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-156889-0
• Package Unit: Get quote
• Quantity Unit: STK