CYP1B1 ligand 3, CAS 65823-65-6

Product Description: CYP1B1 ligand 3 (Compound A1) is a selective inhibitor for cytochrome P450 enzyme CYP1B1 with an IC50 of 11.9 nM. CYP1B1 ligand 3 can be utilized for the synthesis of PROTAC CYP1B1 degrader-2 (HY-158429)[1].

Formula: C18H12ClN3S2

References: [1]Yao X, et al., Development of novel N-aryl-2,4-bithiazole-2-amine-based CYP1B1 degraders for reversing drug resistance. Eur J Med Chem. 2024 Jun 5;272:116488.

CAS Number: 65823-65-6

Molecular Weight: 369.89

Research Area: Cancer

Target: Cytochrome P450

• SKU: MEXHY-159006-10
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-159006-10
• Package Unit: 10 mg
• Quantity Unit: STK