DG013A (formate)

Product Description: DG013A (formate) is a phosphinic acid tripeptide mimetic inhibitor. DG013A (formate) displays significantly weak affinity for both ERAP1 (IC50=33 nM) and ERAP2 (IC50=11 nM). DG013A (formate) can be used for the research of autoimmune disease and cancer[1].

Formula: C27H37N4O4P.2/5CH2O2

References: [1]Birgit Wilding, et al. Investigating the phosphinic acid tripeptide mimetic DG013A as a tool compound inhibitor of the M1-aminopeptidase ERAP1. Bioorg Med Chem Lett. 2021 Jun 15;42:128050.

Molecular Weight: 530.99

Compound Purity: 99.60

Research Area: Cancer; Inflammation/Immunology

Target: Aminopeptidase

• SKU: MEXHY-139907B-5
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-139907B-5
• Package Unit: 5 mg
• Quantity Unit: STK