ELB-139, CAS 188116-08-7

Product Description: ELB-139 is a progesterone analogue. ELB-139 is a GABAA receptor partial agonist. ELB-139 has anxiolytic and anticonvulsant activity. ELB-139 induces increase of extracellular 5-HT in the striatum and the medial prefrontal cortex of rats[1][2].

Formula: C14H16ClN3O

References: [1]Rabe H, et al. The novel anxiolytic ELB139 displays selectivity to recombinant GABA(A) receptors different from diazepam. Neuropharmacology. 2007 Mar;52(3):796-801./[2]Langen B, et al. ELB139 an agonist at the benzodiazepine binding site increases 5-HT in the striatum and prefrontal cortex of rats: a microdialysis study. Pharmacol Biochem Behav. 2007 Jan;86(1):79-85.

CAS Number: 188116-08-7

Molecular Weight: 277.75

Research Area: Neurological Disease

Target: GABA Receptor

• SKU: MEXHY-106437-10
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-106437-10
• Package Unit: 10 mg
• Quantity Unit: STK