EPZ011989 (trifluoroacetate), CAS 1598383-41-5

Product Description: EPZ-011989 trifluoroacetate is a potent and orally active Zeste Homolog 2 (EZH2) inhibitor with metabolic stability. EPZ-011989 trifluoroacetate has inhibitory inhibition for EZH2 with a Ki value of [1]. EPZ011989 (trifluoroacetate) is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.

Applications: Neuroscience-Neuromodulation

Formula: C37H52F3N5O6

References: [1]Campbell JE, et al. EPZ011989, A Potent, Orally-Available EZH2 Inhibitor with Robust in Vivo Activity. ACS Med Chem Lett. 2015 Mar 4;6(5):491-495.

CAS Number: 1598383-41-5

Molecular Weight: 719.83

Compound Purity: 98.71

Research Area: Cancer

Solubility: DMSO : 100 mg/mL (ultrasonic)

Target: Histone Methyltransferase

• SKU: MEXHY-16986A-0
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-16986A-0
• Package Unit: Get quote
• Quantity Unit: STK