ERα degrader 12

ERα degrader 12
SKU
MEXHY-170806-0
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Manufacturer
MedChemExpress

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Product Description: ERα degrader 12 (Compound RA3) is an estrogen receptor α (ERα) degrader with antitumor properties. ERα degrader 12 induces pronounced tumor growth inhibition in a breast cancer xenograft mouse model[1].

Applications: Cancer-programmed cell death

Formula: C39H41NO9S

References: [1]Qing L, et al. Discovery of D-Ring-Contracted Artemisinin as a Potent Hydrophobic Tag for Targeted Protein Degradation. J Med Chem. 2025 Jan 23;68(2):1619-1631.

Molecular Weight: 699.81

Research Area: Cancer

Target: Estrogen Receptor/ERR
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SKU MEXHY-170806-0
Manufacturer MedChemExpress
Manufacturer SKU HY-170806-0
Package Unit Get quote
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