GABAA receptor modulator-4

Product Description: GABAA receptor modulator-4 (Compound 4) is the negative allosteric modulator for GABAA receptor. GABAA receptor modulator-4 inhibits α1β3γ2 GABAA receptor-mediated peak and steady currents with IC50 of 10 μM and 10 μM[1].

Formula: C15H17BrO4S

References: [1]Xu Y, et al., Design, Synthesis, and Pharmacological Evaluation of Nonsteroidal Tricyclic Ligands as Modulators of GABAA Receptors. J Med Chem. 2025 Feb 13;68(3):3795-3813.

Molecular Weight: 373.26

Research Area: Neurological Disease

Target: GABA Receptor

• SKU: MEXHY-170902-0
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-170902-0
• Package Unit: Get quote
• Quantity Unit: STK