GGTI-2133, CAS 191102-79-1

Product Description: GGTI-2133 is an inhibitor for geranylgeranyltransferase I (GGTase-I) with an IC50 of 38 nM. GGTI-2133 inhibits the geranylation of Rap-1A with an IC50 of 10 μM[1].

Applications: COVID-19-immunoregulation

Formula: C27H28N4O3

References: [1]Vasudevan A, et al., Potent, highly selective, and non-thiol inhibitors of protein geranylgeranyltransferase-I. J Med Chem. 1999 Apr 22;42(8):1333-40.

CAS Number: 191102-79-1

Molecular Weight: 456.54

Compound Purity: 98.50

Research Area: Inflammation/Immunology

Solubility: DMSO : 100 mg/mL (ultrasonic)

Target: YAP

• SKU: MEXHY-12369-10.1
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-12369-10.1
• Package Unit: 10 mM/1 ml
• Quantity Unit: STK