Product Description: Gintemetostat (KTX-1001) is a potent NSD2 inhibitor with an IC50 ranging from 0.001 μM to 0.01 μM. As a piperidinyl-methyl-purineamine derivative, gintemetostat has potential applications in cancer research[1].
Applications: Cancer-programmed cell death
Formula: C25H26F4N8O2
References: [1]Roberts M F, et al. 6-Methoxyflavonols from Brickellia veronicaefolia (compositae)[J]. Phytochemistry, 1980, 19(1): 127-129.
CAS Number: 2604513-16-6
Molecular Weight: 546.52
Compound Purity: 99.81
Research Area: Cancer
Solubility: DMSO : 100 mg/mL (ultrasonic)
Target: Histone Methyltransferase