GJG057, CAS 2761767-18-2

Product Description: GJG057 is a selective, orally active inhibitor for leukotriene C4 synthase (LTC4S) with an IC50 of 44 nM. GJG057 exhibits anti-inflammatory activity in mouse skin inflammation model and mouse asthma model[1].

Formula: C21H21F5N4O2

References: [1]Thoma G, et al., Discovery of GJG057, a Potent and Highly Selective Inhibitor of Leukotriene C4 Synthase. J Med Chem. 2025 Feb 27;68(4):4721-4742.

CAS Number: 2761767-18-2

Molecular Weight: 456.41

Research Area: Inflammation/Immunology

Target: Glutathione S-transferase

• SKU: MEXHY-168498-0
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-168498-0
• Package Unit: Get quote
• Quantity Unit: STK