PI3Kδ/BET-IN-1, CAS 3054869-10-9

Product Description: PI3Kδ/BET-IN-1 (compound 10b) shows excellent and balanced activities against PI3Kδ (IC50 = 112 nM) and BRD4-BD1 (IC50 = 19 nM) and exhibits strong antiproliferative activities in DLBCL cells[1].

Formula: C27H34N6O3S

References: [1]Kai Ran, et al. Design, Synthesis, and Biological Evaluation of Thieno[3,2-d]pyrimidine Derivatives as the First Bifunctional PI3Kδ Isoform Selective/Bromodomain and Extra-Terminal Inhibitors. J Med Chem. 2025 Jan 24.

CAS Number: 3054869-10-9

Molecular Weight: 522.66

Research Area: Cancer

Target: Epigenetic Reader Domain;PI3K

• SKU: MEXHY-172130-0
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-172130-0
• Package Unit: Get quote
• Quantity Unit: STK