PPARγ modulator-3

PPARγ modulator-3
SKU
MEXHY-176062-0
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MedChemExpress

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Product Description: PPARγ modulator-3 (Compound 11) is a peroxisome proliferator-activated receptor γ (PPARγ) modulator with a KD value of 186 nM. PPARγ modulator-3 is promising for research of insulin resistance (IR)-related diseases, such as type 2 diabetes mellitus (T2DM) and metabolic syndrome[1].

Formula: C18H13BrO6

References: [1]Cazzaniga G, et al. Enhancing the Activity of γ-Hydroxy Lactone Derivatives as Innovative Peroxisome Proliferator-Activated Receptor γ Non-Agonists Inhibiting Cyclin-Dependent Kinase 5-Mediated Phosphorylation[J]. European Journal of Medicinal Chemistry, 2025: 117657.

Molecular Weight: 405.20

Research Area: Metabolic Disease

Target: PPAR
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SKU MEXHY-176062-0
Manufacturer MedChemExpress
Manufacturer SKU HY-176062-0
Package Unit Get quote
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