Product Description: (Rac)-Aurora A/PKC-IN-1 (Compund 2e) is an orally active Aurora A and PKC (α, β1, β2 and θ) kinase inhibitor. (Rac)-Aurora A/PKC-IN-1 has antiproliferative activity in breast cancer cells in vitro and antimetastatic activity in vivo[1].
Formula: C16H14N6OSe2
References: [1]Bijian K, et al. Novel Aurora A and Protein Kinase C (α, β1, β2, and θ) Multitarget Inhibitors: Impact of Selenium Atoms on the Potency and Selectivity. J Med Chem. 2022 Feb 24;65(4):3134-3150.
CAS Number: 2143100-98-3
Molecular Weight: 464.24
Research Area: Cancer
Target: Aurora Kinase;PKC