rel-Erteberel, CAS 533883-77-1

rel-Erteberel, CAS 533883-77-1
SKU
MEXHY-18295A-1
Packaging Unit
1 mg
Manufacturer
MedChemExpress

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Product Description: rel-Erteberel is rel isomer of Erteberel (HY-18295). Erteberel is a potent and selective estrogen receptor beta (ERβ) agonist with Ki and EC50 of 1.54 nM and 3.61 nM, respectively. Erteberel has anti-tumor activities[1][2].

Applications: Neuroscience-Neuromodulation

Formula: C18H18O3

References: [1]Zhao L, et al. Pharmacological activation of estrogen receptor beta augments innate immunity to suppress cancer metastasis. Proc Natl Acad Sci U S A. 2018 Apr 17;115(16):E3673-E3681./[2]Sareddy GR, et al. Selective Estrogen Receptor β Agonist LY500307 as a Novel Therapeutic Agent for Glioblastoma. Sci Rep. 2016 Apr 29;6:24185.

CAS Number: 533883-77-1

Molecular Weight: 282.33

Research Area: Neurological Disease

Solubility: 10 mM in DMSO

Target: Estrogen Receptor/ERR
More Information
SKU MEXHY-18295A-1
Manufacturer MedChemExpress
Manufacturer SKU HY-18295A-1
Package Unit 1 mg
Quantity Unit STK
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