SCP1-IN-2, CAS 2764615-56-5

Product Description: SCP1-IN-2 (Compound SH T-65) is a potent and selective covalent inhibitor against SCP1. SCP1-IN-2 promotes REST degradation and reduces transcriptional activity. A high level of REST protein drives the tumor growth in some glioblastoma cells. SCP1-IN-2 has the potential for the research of glioblastoma whose growth is driven by REST transcription activity[1].

Applications: Cancer-programmed cell death

Formula: C19H17F3N2O6S2

References: [1]Medellin B, et al. Targeted Covalent Inhibition of Small CTD Phosphatase 1 to Promote the Degradation of the REST Transcription Factor in Human Cells. J Med Chem. 2022;65(1):507-519.

CAS Number: 2764615-56-5

Molecular Weight: 490.47

Compound Purity: 98.77

Research Area: Cancer; Neurological Disease

Solubility: DMSO : 100 mg/mL (ultrasonic)

Target: Phosphatase

• SKU: MEXHY-142683-1
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-142683-1
• Package Unit: 1 mg
• Quantity Unit: STK