SR-1277, CAS 1446715-47-4

Product Description: SR-1277 is a potent, selective and ATP competitive CK1δ/ε inhibitor, with IC50s of 49 nM and 260 nM, respectively. SR-1277 also inhibits FLT3, CDK4/cyclin D1, CDK6/cyclin D3 and CDK9/cyclin K, with IC50s of 305 nM, 1340 nM, 311 nM and 109 nM, respectively. SR-1277 can be used for the research of cancer[1].

Applications: Cancer-Kinase/protease

Formula: C21H19N9O3S

References: [1]Bibian M, et, al. Development of highly selective casein kinase 1δ/1ε (CK1δ/ε) inhibitors with potent antiproliferative properties. Bioorg Med Chem Lett. 2013 Aug 1;23(15):4374-80.

CAS Number: 1446715-47-4

Molecular Weight: 477.50

Research Area: Cancer

Solubility: 10 mM in DMSO

Target: Casein Kinase

• SKU: MEXHY-108907-10
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-108907-10
• Package Unit: 10 mg
• Quantity Unit: STK