VU0810464, CAS 2126040-21-7

Shelf life (days): 1460

Info: A GIRK1/2 and GIRK1/4 activator; induces GIRK1/2 and GIRK1/4 activity in a thallium flux assay using HEK293 cells expressing GIRK1 and GIRK2 or GIRK1 and GIRK4 (EC50s = 165 and 720 nM, respectively); reduces stress-induced hyperthermia at 10 and 30 mg/kg, i.p. in mice but does not affect the percentage of time spent or distance traveled in the open arms of the elevated plus maze in mice at 30 mg/kg

Formulation: A solid

Formal Name: 3-chloro-N-(1-cyclohexyl-3-methyl-1H-pyrazol-5-yl)-4-fluoro-benzeneacetamide

Purity: ≥98%

Formula Markup: C18H21ClFN3O

Formula Weight: 349.834403

CAS Number: 2126040-21-7

• SKU: CAY43073-10
• Manufacturer: Cayman Chemical
• Manufacturer SKU: 43073-10
• Package Unit: 10 mg
• Quantity Unit: STK