ZEN-3411, CAS 1952264-36-6

Product Description: ZEN-3411 is a BET inhibitor with IC50s of 0.05, 0.05 and 0.06 μM for BRD4(BD1), BRD4(BD2) and BRD4(BD1BD2), respectively. ZEN-3411 can be used to form PROTACs to induce degradation of BRD4[1].

Applications: Cancer-programmed cell death

Formula: C21H20N4O2

References: [1]Kharenko OA, et al. Design and Characterization of Novel Covalent Bromodomain and Extra-Terminal Domain (BET) Inhibitors Targeting a Methionine. J Med Chem. 2018 Sep 27;61(18):8202-8211.

CAS Number: 1952264-36-6

Molecular Weight: 360.41

Research Area: Cancer

Solubility: 10 mM in DMSO

Target: Epigenetic Reader Domain

• SKU: MEXHY-111979-1
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-111979-1
• Package Unit: 1 mg
• Quantity Unit: STK